SCHEMBL4603770

SCHEMBL4603770

CC(=O)C(=O)OC(COC(=O)CC[C@H](Nc1ccccc1)C(=O)O)CO[N+](=O)[O-]

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.41
PTGS1 P23219 2/20 0.36
CYP1A2 P05177 2/20 0.32
CYP2C19 P33261 2/20 0.32
GAA P10253 1/20 0.31
ALDH1A1 P00352 2/20 0.31
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
HPGD P15428 1/20 0.31
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30
MMP8 P22894 1/20 0.30
MMP12 P39900 1/20 0.30
MMP14 P50281 1/20 0.30
KEAP1 Q14145 1/20 0.30
DRD4 P21917 1/20 0.30
SLC6A2 P23975 1/20 0.30
CCKAR P32238 1/20 0.30
OPRM1 P35372 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4587980 0.78 PTGS2 (0.37) PTGS2PTGS1CYP1A2ALDH1A1KMT2A
SCHEMBL5278808 0.73 MEN1 (0.40) CYP1A2CYP2C19ALDH1A1KMT2AMEN1
SCHEMBL4585809 0.71 PTGS2 (0.48) PTGS2PTGS1ALDH1A1
SCHEMBL4587179 0.69 PTGS2 (0.37) PTGS2PTGS1CYP1A2CYP2C19ALDH1A1
SCHEMBL4847471 0.68 ALDH1A1 (0.35) PTGS2PTGS1CYP1A2CYP2C19GAA
SCHEMBL30818291 0.68 GAA (0.48) GAAALDH1A1KMT2AHPGDMMP2
SCHEMBL60370 0.65 GAA (0.62) GAAKMT2AMMP9MMP8KEAP1
SCHEMBL60371 0.65 GAA (0.62) GAAKMT2AMMP9MMP8KEAP1
SCHEMBL4587072 0.64 MAPT (0.38) PTGS2ALDH1A1
SCHEMBL2235690 0.64 ALDH1A1 (0.44) GAAALDH1A1KMT2AMEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1692107-A4 NITRIC OXIDE RELEASING PYRUVATE COMPOUNDS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-10-29 EP claimed
EP-1692107-A2 NITRIC OXIDE RELEASING PYRUVATE COMPOUNDS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2006-08-23 EP claimed
WO-2005060603-A2 NITRIC OXIDE RELEASING PYRUVATE COMPOUNDS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2005-07-07 WO claimed