SCHEMBL4604234

SCHEMBL4604234

CCCc1ccc(OCCOc2c(C(=O)C(C)(C)C)sc3ccccc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 2/20 0.56
MAPT P10636 4/20 0.43
ALDH1A1 P00352 3/20 0.43
LMNA P02545 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
CNR2 P34972 1/20 0.42
NPC1 O15118 3/20 0.41
KMT2A Q03164 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.39
PPARG P37231 3/20 0.39
PPARD Q03181 2/20 0.39
PPARA Q07869 2/20 0.39
S1PR4 O95977 1/20 0.39
S1PR1 P21453 1/20 0.39
S1PR3 Q99500 1/20 0.39
S1PR5 Q9H228 1/20 0.39
BCL2 P10415 1/20 0.39
BCL2L1 Q07817 1/20 0.39
MCL1 Q07820 1/20 0.39
BAD Q92934 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4828979 0.89 CXCR2 (0.57) CXCR2LMNAL3MBTL1PPARGPPARD
SCHEMBL4604550 0.87 CXCR2 (0.59) CXCR2MAPTALDH1A1LMNARXFP1
SCHEMBL4606075 0.84 CXCR2 (0.61) CXCR2MAPTALDH1A1LMNARXFP1
SCHEMBL4602716 0.77 CXCR2 (0.54) CXCR2MAPTALDH1A1LMNARXFP1
SCHEMBL4604985 0.77 CXCR2 (0.54) CXCR2MAPTLMNAKMT2AL3MBTL1
SCHEMBL4604246 0.76 CXCR2 (0.53) CXCR2MAPTALDH1A1LMNARXFP1
SCHEMBL4633571 0.75 CXCR2 (0.55) CXCR2MAPTALDH1A1LMNARXFP1
SCHEMBL4606183 0.75 CXCR2 (0.48) CXCR2MAPTALDH1A1LMNAKMT2A
SCHEMBL4605238 0.75 CXCR2 (0.52) CXCR2MAPTALDH1A1LMNARXFP1
SCHEMBL4633030 0.74 CXCR2 (0.52) CXCR2LMNAL3MBTL1PPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685122-B1 BENZOFURANS AND BENZOTHIOPHENES MERCK PATENT GMBH (DE) 2008-07-09 EP disclosed