SCHEMBL4605555

SCHEMBL4605555

CC(O)C(Oc1cccc2[nH]c3ccccc3c12)N1CCN(CC2CC2)CC1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 16/20 0.49
ADRB2 P07550 11/20 0.48
ADRB1 P08588 11/20 0.48
DNM1 Q05193 1/20 0.42
DRD1 P21728 1/20 0.40
DRD5 P21918 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4607514 0.85 ADRB3 (0.49) ADRB3ADRB2ADRB1DNM1
SCHEMBL4605132 0.82 ADRB3 (0.46) ADRB3ADRB2ADRB1DNM1DRD1
SCHEMBL4606756 0.80 ADRB3 (0.47) ADRB3ADRB2ADRB1DNM1
SCHEMBL2983464 0.80 ADRB3 (0.74) ADRB3ADRB2ADRB1DNM1
SCHEMBL4607708 0.79 BCHE (0.46) ADRB3ADRB2ADRB1DNM1DRD1
SCHEMBL4606968 0.78 ADRB3 (0.42) ADRB3ADRB2ADRB1DNM1
SCHEMBL4607757 0.76 POLB (0.44) ADRB3ADRB2ADRB1DNM1
SCHEMBL4607185 0.76 ADRB3 (0.46) ADRB3ADRB2ADRB1DNM1
SCHEMBL4608603 0.75 ADRB3 (0.49) ADRB3ADRB2ADRB1
SCHEMBL4607629 0.74 KDM4E (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP claimed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO claimed