SCHEMBL4607708

SCHEMBL4607708

COc1cc(OC)c(CN2CCN(C(Oc3cccc4[nH]c5ccccc5c34)C(C)O)CC2)c(OC)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.46
CHRNB2 P17787 1/20 0.46
ACHE P22303 1/20 0.46
CHRNA7 P36544 1/20 0.46
CHRNA4 P43681 1/20 0.46
ADRB3 P13945 9/20 0.45
ADRB2 P07550 9/20 0.45
ADRB1 P08588 7/20 0.45
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
DRD2 P14416 3/20 0.39
TLR4 O00206 2/20 0.39
DNM1 Q05193 2/20 0.39
KDM4E B2RXH2 1/20 0.39
SLC22A2 O15244 1/20 0.39
SLC22A1 O15245 1/20 0.39
MLNR O43193 1/20 0.39
NR1I2 O75469 1/20 0.39
KCNK2 O95069 1/20 0.39
ABCB11 O95342 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4606756 0.90 ADRB3 (0.47) BCHECHRNB2ACHECHRNA7CHRNA4
SCHEMBL4607514 0.84 ADRB3 (0.49) BCHECHRNB2ACHECHRNA7CHRNA4
SCHEMBL2993358 0.83 ADRB2 (0.65) BCHECHRNB2ACHECHRNA7CHRNA4
SCHEMBL4605555 0.79 ADRB3 (0.49) ADRB3ADRB2ADRB1DNM1DRD1
SCHEMBL4605132 0.77 ADRB3 (0.46) ADRB3ADRB2ADRB1KMT2ADRD2
SCHEMBL4608053 0.77 MAPT (0.50) ADRB3ADRB2ADRB1KMT2AMEN1
SCHEMBL4605749 0.76 TLR9 (0.49) ADRB3ADRB2ADRB1KDM4EGAA
SCHEMBL4607757 0.75 POLB (0.44) BCHECHRNB2ACHECHRNA7CHRNA4
SCHEMBL4606968 0.74 ADRB3 (0.42) ADRB3ADRB2ADRB1KMT2AMEN1
SCHEMBL2994599 0.73 ADRB2 (0.68) ADRB3ADRB2ADRB1KMT2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP claimed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO claimed
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP disclosed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO disclosed