SCHEMBL4607185

SCHEMBL4607185

CC(O)C(Oc1cccc2[nH]c3ccccc3c12)N1CCN(C(=O)Cc2ccc(F)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 6/20 0.46
ADRB2 P07550 6/20 0.46
ADRB1 P08588 5/20 0.46
MAPT P10636 4/20 0.41
HSD17B10 Q99714 3/20 0.41
POLB P06746 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 3/20 0.39
HPGD P15428 1/20 0.39
HRH3 Q9Y5N1 2/20 0.39
DNM1 Q05193 1/20 0.39
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4608053 0.91 MAPT (0.50) ADRB3ADRB2ADRB1MAPTHSD17B10
SCHEMBL4607632 0.90 MET (0.41) ADRB3ADRB2ADRB1MAPTHSD17B10
SCHEMBL4605834 0.87 CYP1A2 (0.44) ADRB3ADRB2ADRB1MAPTHSD17B10
SCHEMBL4608603 0.86 ADRB3 (0.49) ADRB3ADRB2ADRB1KDM4EALDH1A1
SCHEMBL4606968 0.85 ADRB3 (0.42) ADRB3ADRB2ADRB1MAPTHSD17B10
SCHEMBL2993325 0.80 ADRB3 (0.67) ADRB3ADRB2ADRB1DNM1
SCHEMBL4605132 0.80 ADRB3 (0.46) ADRB3ADRB2ADRB1MAPTKDM4E
SCHEMBL4607629 0.79 KDM4E (0.52) MAPTHSD17B10L3MBTL1KDM4EALDH1A1
SCHEMBL4607514 0.78 ADRB3 (0.49) ADRB3ADRB2ADRB1KDM4EDNM1
SCHEMBL4608607 0.78 ALDH1A1 (0.44) ADRB3ADRB2ADRB1HSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP claimed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO claimed
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP disclosed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO disclosed