SCHEMBL4606166

SCHEMBL4606166

Cc1ccc(-c2nc(CCNCC(=O)N3CCCC3)c[nH]2)nc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.40
DPP4 P27487 1/20 0.40
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
JAK3 P52333 1/20 0.36
GRIN2B Q13224 3/20 0.36
ALDH1A1 P00352 2/20 0.36
HSD17B10 Q99714 1/20 0.36
SMO Q99835 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4603052 0.80 DGAT2 (0.38) CYP2D6DPP4GRIN2BHSD17B10HPGD
SCHEMBL4605631 0.80 PRMT3 (0.43) CYP2D6DPP4
SCHEMBL4606161 0.69 ALDH1A1 (0.41) CYP2D6DPP4ALDH1A1HSD17B10HPGD
SCHEMBL4605625 0.65 PRMT3 (0.39) CYP2D6DPP4SMN1; SMN2
SCHEMBL4603048 0.65 KMT2A (0.42) CYP2D6ALDH1A1HPGD
SCHEMBL17144250 0.65 CYP2D6 (0.46) CYP2D6DPP4ALDH1A1LMNAHPGD
SCHEMBL13313010 0.62 SMN1; SMN2 (0.57) ALDH1A1LMNAHPGDNPC1RAB9A
SCHEMBL2646670 0.61 DPP4 (0.50) CYP2D6DPP4ALDH1A1LMNAHPGD
SCHEMBL28509553 0.61 ALDH1A1 (0.67) ALDH1A1HSD17B10LMNAHPGDNPC1
SCHEMBL10677073 0.60 IDO1 (0.35) GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917001-A2 PHARMACEUTICAL COMPOSITION COMPRISING A DPP-IV INHIBITOR F.HOFFMANN-LA ROCHE AG (CH) 2008-05-07 EP disclosed
WO-2007017423-A2 PHARMACEUTICAL COMPOSITION COMPRISING A DPP-IV INHIBITOR F. HOFFMANN-LA ROCHE AG (CH) 2007-02-15 WO disclosed