SCHEMBL4606348

SCHEMBL4606348

O=C(Cc1ccsc1)N[C@@H](CCCSCC(=O)C(F)(F)F)C(=O)Nc1cc(Cl)cc(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.39
MARS1 P56192 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
GLS O94925 2/20 0.34
RAB9A P51151 2/20 0.34
KMT2A Q03164 2/20 0.34
NPC1 O15118 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
MEN1 O00255 1/20 0.33
CES1 P23141 1/20 0.33
FABP4 P15090 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4605614 0.87 CES1 (0.45) RAB9AKMT2AHDAC1HDAC2MEN1
SCHEMBL4166185 0.85 NPC1 (0.42) POLBRAB9AKMT2ANPC1TDP1
Trifluoroacetic Acid SCHEMBL4169498 0.83 HDAC4 (0.39) L3MBTL1HDAC1HDAC2
SCHEMBL4174445 0.81 HDAC1 (0.42) POLBRAB9AKMT2ANPC1HDAC1
Trifluoroacetic Acid SCHEMBL4160622 0.81 PADI4 (0.39) POLBGLSHDAC1HDAC2CES1
SCHEMBL4174424 0.81 SIGMAR1 (0.38) L3MBTL1KMT2AHDAC1HDAC2MEN1
SCHEMBL4605724 0.80 CES1 (0.46) HDAC1HDAC2CES1
SCHEMBL4164039 0.78 HDAC1 (0.41) POLBKMT2AHDAC1HDAC2MEN1
Trifluoroacetic Acid SCHEMBL4166937 0.78 FABP4 (0.36) KMT2AHDAC1HDAC2MEN1CES1
SCHEMBL3507605 0.77 GPR139 (0.42) L3MBTL1KMT2AHDAC1HDAC2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945609-A2 AMINO ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2008-07-23 EP disclosed
WO-2007029036-A2 AMINO ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2007-03-15 WO disclosed