SCHEMBL4607079

SCHEMBL4607079

CC(C)S(=O)(=O)N[C@H]1CCC[C@H]1c1ccc(NC(=O)c2cccc(NC(=O)OC(C)(C)C)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 13/20 0.49
GRIA2 P42262 4/20 0.48
KAT6A Q92794 1/20 0.43
KCNH2 Q12809 2/20 0.42
KDM1A O60341 1/20 0.42
MAOA P21397 1/20 0.42
KDM1B Q8NB78 1/20 0.42
RCOR1 Q9UKL0 1/20 0.42
PRMT5 O14744 1/20 0.41
WDR77 Q9BQA1 1/20 0.41
STAT3 P40763 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4607349 0.91 GRIA4 (0.54) GRIA4GRIA2KDM1ARCOR1
SCHEMBL4605831 0.87 GRIA4 (0.55) GRIA4GRIA2KCNH2
SCHEMBL4605833 0.87 GRIA4 (0.55) GRIA4GRIA2KCNH2
SCHEMBL4606805 0.84 GRIA4 (0.55) GRIA4GRIA2KCNH2
SCHEMBL4607636 0.84 GRIA4 (0.57) GRIA4GRIA2KCNH2
SCHEMBL4607477 0.84 GRIA4 (0.57) GRIA4GRIA2KCNH2
SCHEMBL4605829 0.83 GRIA4 (0.56) GRIA4GRIA2KCNH2KDM1AMAOA
SCHEMBL4607371 0.83 GRIA4 (0.56) GRIA4GRIA2KCNH2KDM1AMAOA
SCHEMBL4607600 0.82 GRIA4 (0.70) GRIA4GRIA2KDM1AMAOAKDM1B
SCHEMBL4607075 0.82 GRIA4 (0.70) GRIA4GRIA2KDM1AMAOAKDM1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246797-B1 CYCLOPENTYL SULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2008-07-23 EP claimed
EP-1246797-B1 CYCLOPENTYL SULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2008-07-23 EP disclosed