SCHEMBL4607143

SCHEMBL4607143

CCCC(F)OC(=O)Nc1cccc(C#N)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.49
PDK2 Q15119 1/20 0.49
PDK3 Q15120 1/20 0.49
PDK4 Q16654 1/20 0.49
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 2/20 0.49
MAPT P10636 2/20 0.49
MEN1 O00255 1/20 0.49
LMNA P02545 1/20 0.48
MCHR1 Q99705 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
RXFP1 Q9HBX9 1/20 0.46
MAPK1 P28482 1/20 0.45
HSD17B10 Q99714 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
HTT P42858 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
TSHR P16473 1/20 0.44
GRM4 Q14833 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27641762 0.81 LMNA (0.47) PDK1PDK2PDK3PDK4KMT2A
SCHEMBL19592329 0.78 HSD17B10 (0.67) PDK1PDK2PDK3PDK4KMT2A
SCHEMBL4598556 0.78 MAPT (0.62) PDK1PDK2PDK3PDK4KMT2A
SCHEMBL6130895 0.76 KDM4E (0.43) KMT2AALDH1A1MAPTMEN1LMNA
SCHEMBL6130860 0.76 HPGD (0.47) KMT2AALDH1A1MAPTMEN1LMNA
SCHEMBL15219819 0.75 SMN1; SMN2 (0.49) PDK1PDK2PDK3PDK4KMT2A
SCHEMBL12989323 0.75 MAPT (0.65) PDK1PDK2PDK3PDK4KMT2A
SCHEMBL12330810 0.75 SMN1; SMN2 (0.47) PDK1PDK2PDK3PDK4KMT2A
SCHEMBL3860997 0.75 CTSL (0.47) PDK1PDK2PDK3PDK4KMT2A
SCHEMBL4599065 0.74 LMNA (0.63) PDK1PDK2PDK3PDK4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948624-A2 PROCESS FOR THE PREPARATION OF BENZO[E][1,2,4]TRIAZEPIN-2-ONE DERIVATIVES Janssen Pharmaceutica, N.V. (BE) 2008-07-30 EP disclosed
WO-2007035430-A2 PROCESS FOR THE PREPARATION OF BENZO [E] [1,2,4] TRIAZEPIN-2-ONE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 2007-03-29 WO disclosed