SCHEMBL4607534

SCHEMBL4607534

CC(CCC=O)Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
KCNH2 Q12809 3/20 0.40
TMEM97 Q5BJF2 3/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
P2RX3 P56373 1/20 0.38
TAAR1 Q96RJ0 1/20 0.37
PPARG P37231 3/20 0.36
PPARA Q07869 3/20 0.36
EPHX2 P34913 1/20 0.36
IDO1 P14902 1/20 0.36
SLC6A9 P48067 1/20 0.36
FDFT1 P37268 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19407026 0.80 ALDH1A1 (0.44) ALDH1A1KCNH2TMEM97NPC1RAB9A
SCHEMBL11611907 0.78 ALDH1A1 (0.42) ALDH1A1KCNH2TMEM97NPC1RAB9A
SCHEMBL15865878 0.78 ITGB1 (0.36) ALDH1A1TP53TSHRNPC1RAB9A
SCHEMBL7925119 0.78 TAAR1 (0.50) NPC1RAB9AMEN1KMT2ATAAR1
SCHEMBL28185303 0.77 ALDH1A1 (0.41) ALDH1A1KCNH2TMEM97NPC1RAB9A
SCHEMBL4608415 0.77 ALDH1A1 (0.41) ALDH1A1KCNH2TMEM97NPC1RAB9A
SCHEMBL13971048 0.76 FFAR1 (0.50) PPARGPPARAEPHX2SLC6A9L3MBTL1
SCHEMBL25215174 0.76 TP53 (0.71) ALDH1A1TP53TSHRKCNH2TMEM97
SCHEMBL25252393 0.76 TP53 (0.71) ALDH1A1TP53TSHRKCNH2TMEM97
SCHEMBL16379333 0.76 TP53 (0.71) ALDH1A1TP53TSHRKCNH2TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948603-A1 TETRAHYDROINDOLE DERIVATIVES FOR TREATMENT OF ALZHEIMER'S DISEASE MERCK SHARP & DOHME LTD. (GB) 2008-07-30 EP disclosed
WO-2007054739-A1 TETRAHYDROINDOLE DERIVATIVES FOR TREATMENT OF ALZHEIMER'S DISEASE MERCK SHARP & DOHME LIMITED (GB) 2007-05-18 WO disclosed