SCHEMBL4607673

SCHEMBL4607673

O=C([CH]CCCSCC(=O)C(F)(F)F)NCc1ccco1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
HPGD P15428 6/20 0.48
POLB P06746 5/20 0.48
L3MBTL1 Q9Y468 4/20 0.48
MAPT P10636 2/20 0.48
KDM4E B2RXH2 1/20 0.48
PTPN7 P35236 1/20 0.48
HSD17B10 Q99714 1/20 0.48
MLYCD O95822 1/20 0.47
TDP1 Q9NUW8 2/20 0.46
APEX1 P27695 1/20 0.46
RECQL P46063 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
EPHX2 P34913 3/20 0.44
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.42
CES1 P23141 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4607677 0.82 HPGD (0.62) ALDH1A1HPGDPOLBL3MBTL1MAPT
SCHEMBL4606734 0.73 NPY1R (0.46) ALDH1A1HPGDPOLBL3MBTL1MAPT
SCHEMBL7415087 0.71 MLYCD (0.64) ALDH1A1HPGDPOLBL3MBTL1MAPT
SCHEMBL4169539 0.70 MAPT (0.41) ALDH1A1HPGDPOLBL3MBTL1MAPT
SCHEMBL28017807 0.69 POLB (0.65) ALDH1A1HPGDPOLBL3MBTL1MAPT
SCHEMBL4156245 0.69 CES1 (0.44) ALDH1A1HPGDPOLBL3MBTL1MAPT
SCHEMBL9420448 0.68 POLB (0.63) ALDH1A1HPGDPOLBL3MBTL1MAPT
SCHEMBL12466814 0.67 MLYCD (0.58) ALDH1A1HPGDPOLBL3MBTL1MAPT
SCHEMBL10320562 0.66 CES1 (0.50) ALDH1A1HPGDPOLBMAPTMLYCD
SCHEMBL2115850 0.66 HPGD (1.00) ALDH1A1HPGDPOLBL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945609-A2 AMINO ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2008-07-23 EP disclosed
WO-2007029036-A2 AMINO ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2007-03-15 WO disclosed