SCHEMBL4607790

SCHEMBL4607790

COC(=O)C(CC(=O)O)Cc1ccc(N)cc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CPA1 P15085 2/20 0.47
CPB1 P15086 1/20 0.47
CPA3 P15088 1/20 0.47
CPB2 Q96IY4 1/20 0.47
POLB P06746 1/20 0.46
LTA4H P09960 2/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.43
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MMEL1 Q495T6 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3965849 0.86 ESR1 (0.58) CPA1CPB1CPA3CPB2POLB
SCHEMBL2398335 0.85 CPA1 (0.66) CPA1CPB1CPA3CPB2LTA4H
SCHEMBL1914987 0.85 CPA1 (0.66) CPA1CPB1CPA3CPB2LTA4H
SCHEMBL901408 0.85 CPA1 (0.66) CPA1CPB1CPA3CPB2LTA4H
SCHEMBL7365956 0.84 POLB (0.62) CPA1CPB1CPA3CPB2POLB
SCHEMBL3664929 0.84 KMT2A (0.59) CPA1CPB1CPA3CPB2POLB
SCHEMBL16798224 0.84 MMP2 (0.51) CPA1CPB1CPA3CPB2POLB
SCHEMBL14571476 0.84 KMT2A (0.68) POLBLTA4HKMT2AMEN1ALDH1A1
SCHEMBL1912582 0.83 MMEL1 (0.60) CPA1CPB1CPA3CPB2LTA4H
SCHEMBL11586603 0.82 CPA1 (0.70) CPA1CPB1CPA3CPB2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1440976-B1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production BOEHRINGER INGELHEIM PHARMA (DE) 2008-07-23 EP disclosed
EP-1440976-A1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production Boehringer Ingelheim Pharma GmbH & Co.KG (DE) 2004-07-28 EP disclosed
EP-0927192-B1 MODIFIED AMINOACIDS, PHARMACEUTICALS CONTAINING THESE COMPOUNDS AND METHOD FOR THEIR PRODUCTION BOEHRINGER INGELHEIM PHARMA (DE) 2004-05-12 EP disclosed
CN-1129605-C Modified aminoacids, pharmaceuticals containing these compounds and method for their prodn. THOMAE GMBH DR K (DE) 2003-12-03 CN disclosed
CN-1230196-A Modified aminoacids, pharmaceuticals containing these compounds and method for their prodn. THOMAE GMBH DR K (DE) 1999-09-29 CN disclosed