SCHEMBL7365956

SCHEMBL7365956

COC(=O)C(CC(=O)O)Cc1ccc(OC)cc1

nearest known ligand 0.70

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.62
LDHA P00338 1/20 0.58
MMP1 P03956 1/20 0.55
MMP2 P08253 1/20 0.55
MMP3 P08254 1/20 0.55
MMP9 P14780 1/20 0.55
ALDH1A1 P00352 1/20 0.53
KMT2A Q03164 1/20 0.52
PPARG P37231 1/20 0.50
FFAR1 O14842 2/20 0.49
EPHX2 P34913 1/20 0.48
CPA1 P15085 2/20 0.47
CPB1 P15086 1/20 0.47
CPA3 P15088 1/20 0.47
CPB2 Q96IY4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6178867 0.87 LDHA (0.67) POLBLDHAMMP1MMP2MMP3
SCHEMBL3965849 0.86 ESR1 (0.58) POLBKMT2ACPA1CPB1CPA3
SCHEMBL1914987 0.85 CPA1 (0.66) MMP2MMP9KMT2ACPA1CPB1
SCHEMBL901408 0.85 CPA1 (0.66) MMP2MMP9KMT2ACPA1CPB1
SCHEMBL2398335 0.85 CPA1 (0.66) MMP2MMP9KMT2ACPA1CPB1
SCHEMBL16798224 0.84 MMP2 (0.51) POLBMMP2MMP9KMT2APPARG
SCHEMBL3664929 0.84 KMT2A (0.59) POLBALDH1A1KMT2APPARGEPHX2
SCHEMBL4607790 0.84 CPA1 (0.47) POLBALDH1A1KMT2ACPA1CPB1
SCHEMBL28201178 0.84 EPHX2 (0.64) POLBLDHAKMT2APPARGEPHX2
SCHEMBL10441763 0.83 LTA4H (0.64) PPARGFFAR1CPA1CPB1CPA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242600-B1 ANTIISCHEMIC AGENTS, ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-06-05 US disclosed
EP-0970071-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2000-01-12 EP disclosed
WO-1998039324-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-11 WO disclosed
EP-0217286-A1 Phenylalanine derivative and proteinase inhibitor Okamoto, Shosuke (JP) 1987-04-08 EP disclosed