SCHEMBL4608418

SCHEMBL4608418

CC(C)CC1CC(C(=O)O)CCN1c1nccc(Cl)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PANK3 Q9H999 1/20 0.41
KDM4E B2RXH2 7/20 0.40
CYP2C19 P33261 1/20 0.40
LMNA P02545 2/20 0.37
HTT P42858 1/20 0.37
MMP2 P08253 1/20 0.36
HSD17B10 Q99714 3/20 0.36
HPGD P15428 2/20 0.36
USP2 O75604 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
NEK2 P51955 2/20 0.35
ALDH1A1 P00352 3/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
NOTUM Q6P988 3/20 0.33
RORC P51449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4608417 0.72 LMNA (0.34) PANK3KDM4ECYP2C19LMNAHTT
SCHEMBL3531018 0.71 PANK3 (0.49) PANK3KDM4ECYP2C19LMNAHSD17B10
SCHEMBL12289389 0.67 CYP3A4 (0.50) PANK3KDM4ECYP2C19LMNAHSD17B10
SCHEMBL3783886 0.65 RORC (0.40) KDM4ENEK2ALDH1A1MAPK1KMT2A
SCHEMBL18166973 0.64 PANK3 (0.46) PANK3KDM4ECYP2C19LMNAHTT
SCHEMBL1976029 0.63 KDM4E (0.68) KDM4ECYP2C19LMNAHTTHSD17B10
SCHEMBL4031515 0.63 KDM4E (0.59) KDM4ECYP2C19LMNAHSD17B10HPGD
SCHEMBL27717820 0.63 DYRK1A (0.51) MMP2ALDH1A1
SCHEMBL580419 0.62 RAB9A (0.37) LMNAHSD17B10HPGDNPSR1ALDH1A1
SCHEMBL31402771 0.62 SMO (0.50) PANK3KDM4ECYP2C19LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877385-A1 PYRIMIDINES AND PYRAZINES USEFUL AS MODULATORS OF ION CHANNELS Vertex Pharmaceuticals Incorporated (US) 2008-01-16 EP disclosed
WO-2006119451-A1 PYRIMIDINES AND PYRAZINES USEFUL AS MODULATORS OF ION CHANNELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-11-09 WO disclosed