SCHEMBL4608622

SCHEMBL4608622

O=C(O)Cc1ccc(Cl)cc1CO

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.56
KEAP1 Q14145 1/20 0.50
NFE2L2 Q16236 1/20 0.50
CXCL8 P10145 1/20 0.46
CYP2C9 P11712 1/20 0.46
CHRM1 P11229 1/20 0.46
GRIK1 P39086 1/20 0.43
PTGDR2 Q9Y5Y4 3/20 0.42
LMNA P02545 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TDP1 Q9NUW8 2/20 0.40
PTGDR Q13258 1/20 0.40
CAMK2A Q9UQM7 1/20 0.40
AKR1B1 P15121 1/20 0.39
MEN1 O00255 1/20 0.39
SLC22A1 O15245 1/20 0.39
USP2 O75604 1/20 0.39
HSP90AA1 P07900 1/20 0.39
CYP3A4 P08684 1/20 0.39
HSPD1 P10809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16041940 0.90 KEAP1 (0.54) MAPTKEAP1NFE2L2CXCL8CYP2C9
SCHEMBL28071595 0.83 MAPT (0.50) MAPTCYP2C9LMNAALDH1A1TDP1
SCHEMBL1154758 0.81 IDO1 (0.50) MAPTCYP2C9LMNAALDH1A1TDP1
SCHEMBL29493203 0.81 IDO1 (0.50) MAPTCYP2C9LMNAALDH1A1TDP1
Hydrochloric Acid SCHEMBL3051125 0.80 IDO1 (0.47) MAPTKEAP1NFE2L2CXCL8CYP2C9
SCHEMBL2394432 0.80 KEAP1 (0.53) MAPTKEAP1NFE2L2CXCL8CYP2C9
SCHEMBL260512 0.80 CHRM1 (0.57) KEAP1NFE2L2CXCL8CYP2C9CHRM1
SCHEMBL29419329 0.80 CHRM1 (0.57) KEAP1NFE2L2CXCL8CYP2C9CHRM1
SCHEMBL29497752 0.80 CXCL8 (0.57) MAPTKEAP1NFE2L2CXCL8CYP2C9
SCHEMBL2578143 0.80 CXCL8 (0.57) MAPTKEAP1NFE2L2CXCL8CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948630-A2 NOVEL COMPOUNDS AstraZeneca AB (SE) 2008-07-30 EP disclosed
WO-2007052023-A2 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2007-05-10 WO disclosed