SCHEMBL4609149

SCHEMBL4609149

CCC(C)(O)C(=O)Nc1ccc(S(=O)(=O)c2ccccc2)cc1Cl

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.55
PDK1 Q15118 14/20 0.53
PDK2 Q15119 14/20 0.53
PDK3 Q15120 14/20 0.53
PDK4 Q16654 14/20 0.53
ABCC9 O60706 1/20 0.50
ABCC8 Q09428 1/20 0.50
KCNJ11 Q14654 1/20 0.50
KCNJ8 Q15842 1/20 0.50
NR1H2 P55055 1/20 0.48
NR1H3 Q13133 1/20 0.48
PTGES2 Q9H7Z7 1/20 0.47
LMNA P02545 1/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4609528 0.89 ABCB11 (0.53) ABCB11PDK1PDK2PDK3PDK4
SCHEMBL6570069 0.88 PDK1 (0.60) ABCB11PDK1PDK2PDK3PDK4
SCHEMBL6571101 0.86 PDK1 (0.56) ABCB11PDK1PDK2PDK3PDK4
SCHEMBL4608658 0.85 ABCB11 (0.58) ABCB11PDK1PDK2PDK3PDK4
SCHEMBL4609857 0.83 PDK1 (0.74) ABCB11PDK1PDK2PDK3PDK4
SCHEMBL4609853 0.83 PDK1 (0.74) ABCB11PDK1PDK2PDK3PDK4
SCHEMBL4608406 0.83 PDK1 (0.74) ABCB11PDK1PDK2PDK3PDK4
SCHEMBL4609323 0.82 PDK1 (0.55) ABCB11PDK1PDK2PDK3PDK4
SCHEMBL8866487 0.81 ABCC9 (0.67) ABCC9ABCC8KCNJ11KCNJ8LMNA
SCHEMBL6347588 0.80 PDK1 (0.50) ABCB11PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1059927-B1 CHEMICAL COMPOUNDS AND THEIR USE TO ELEVATE PYRUVATE DEHYDROGENASE ACTIVITY ASTRAZENECA AB (SE) 2008-07-30 EP disclosed