SCHEMBL4609358

SCHEMBL4609358

CCc1ccc(Oc2ccc(C#N)cc2)nc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.53
OPRM1 P35372 1/20 0.52
P2RX3 P56373 6/20 0.47
GAA P10253 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
EGLN1 Q9GZT9 1/20 0.43
KDM4E B2RXH2 2/20 0.43
MAP4K4 O95819 1/20 0.43
RAB9A P51151 1/20 0.43
PGR P06401 1/20 0.43
CYP19A1 P11511 1/20 0.42
LMNA P02545 2/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAOB P27338 1/20 0.41
PDE4B Q07343 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6161241 0.91 OPRM1 (0.58) CYP2A6OPRM1P2RX3GAAL3MBTL1
SCHEMBL4597520 0.85 OPRM1 (0.52) OPRM1P2RX3GAAL3MBTL1EGLN1
SCHEMBL12775734 0.84 OPRM1 (0.49) CYP2A6OPRM1P2RX3GAAL3MBTL1
SCHEMBL19362952 0.81 KDM4E (0.59) P2RX3GAAL3MBTL1EGLN1KDM4E
SCHEMBL15604704 0.80 CYP2A6 (0.76) CYP2A6KDM4ERAB9APGRCYP19A1
SCHEMBL14349927 0.80 P2RX3 (0.48) P2RX3L3MBTL1KDM4EHTTSMN1; SMN2
SCHEMBL27368615 0.80 OPRM1 (0.46) OPRM1P2RX3KDM4EMAP4K4RAB9A
SCHEMBL4598488 0.80 KDM4E (0.50) CYP2A6OPRM1P2RX3GAAKDM4E
SCHEMBL12967186 0.80 MEN1 (0.58) P2RX3L3MBTL1EGLN1KDM4ERAB9A
SCHEMBL12844619 0.79 GRN (0.47) OPRM1L3MBTL1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed