SCHEMBL6161241

SCHEMBL6161241

CCc1ccc(Oc2ccc(C#N)cn2)cc1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.58
CYP2A6 P11509 1/20 0.53
P2RX3 P56373 9/20 0.48
PDE4B Q07343 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
GAA P10253 1/20 0.45
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
HTT P42858 1/20 0.44
MAP4K4 O95819 1/20 0.43
ACACB O00763 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4609358 0.91 CYP2A6 (0.53) OPRM1CYP2A6P2RX3PDE4BL3MBTL1
SCHEMBL3177956 0.85 OPRM1 (0.58) OPRM1P2RX3PDE4BL3MBTL1GAA
SCHEMBL8016836 0.85 OPRM1 (0.58) OPRM1P2RX3PDE4BL3MBTL1GAA
SCHEMBL8237112 0.83 KDM4E (0.54) OPRM1CYP2A6P2RX3PDE4BL3MBTL1
SCHEMBL3692227 0.82 OPRM1 (0.62) OPRM1P2RX3PDE4BL3MBTL1GAA
SCHEMBL5830771 0.82 OPRM1 (0.53) OPRM1P2RX3PDE4BL3MBTL1GAA
SCHEMBL8410055 0.80 OPRM1 (0.57) OPRM1P2RX3PDE4BL3MBTL1GAA
SCHEMBL15604704 0.80 CYP2A6 (0.76) CYP2A6KDM4ERAB9A
SCHEMBL24665295 0.80 OPRM1 (0.52) OPRM1P2RX3PDE4BL3MBTL1HTT
SCHEMBL6160870 0.80 MEN1 (0.58) OPRM1P2RX3PDE4BL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050165064-A1 Novel thiol derivative, process for producing the same and use thereof TAKEDA PHARMACEUTICALS NORTH AMERICA, INC. 2005-07-28 US disclosed
EP-1500658-A1 NOVEL THIOL DERIVATIVE, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2005-01-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050165064-A1 Novel thiol derivative, process for producing the same and use thereof TST, QSOX1, MMP1 OPRM1 2125/4885CYP2A6 587/4885P2RX3 3309/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.