SCHEMBL4610394

SCHEMBL4610394

CN(C)S(=O)(=O)n1cc(CCCc2ccccc2)nc1[Si](C)(C)C(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPSE Q9Y251 1/20 0.35
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
TSHR P16473 1/20 0.33
DAGLA Q9Y4D2 2/20 0.33
ALDH1A1 P00352 1/20 0.33
DHFR P00374 1/20 0.32
POLB P06746 1/20 0.32
AOC3 Q16853 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
GSK3B P49841 1/20 0.31
TLR8 Q9NR97 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22075884 0.87 TSHR (0.35) HPSEMEN1KMT2ATSHRALDH1A1
SCHEMBL2105626 0.73 RIPK1 (0.34)
SCHEMBL22075862 0.66 SMN1; SMN2 (0.41) HPSEMEN1KMT2ATSHRALDH1A1
SCHEMBL7705910 0.66 CA2 (0.32) TSHR
SCHEMBL22075572 0.62 TSHR (0.37) HPSEMEN1KMT2ATSHRALDH1A1
SCHEMBL5816755 0.61 PDE10A (0.50) HPSENOS3NOS1NOS2TSHR
SCHEMBL5326138 0.61 NOS3 (0.49) HPSENOS3NOS1NOS2MEN1
SCHEMBL5303902 0.59 TLR8 (0.48) HPSENOS3NOS1NOS2SIGMAR1
SCHEMBL5814723 0.59 NOS3 (0.43) HPSENOS3NOS1NOS2MEN1
SCHEMBL5305112 0.59 RECQL (0.46) HPSENOS3NOS1NOS2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981880-A2 USE OF 4-IMIDAZOLE DERIVATIVES FOR CNS DISORDERS F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP disclosed
WO-2007085556-A2 USE OF 4-IMIDAZOLE DERIVATIVES FOR CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO disclosed