SCHEMBL4611046

SCHEMBL4611046

CNc1ccc(C)c(-c2ccc(C=CC(=O)O)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.48
NPSR1 Q6W5P4 1/20 0.43
HCAR2 Q8TDS4 2/20 0.42
CA12 O43570 2/20 0.42
AKR1B10 O60218 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA3 P07451 2/20 0.42
AKR1B1 P15121 2/20 0.42
CA4 P22748 2/20 0.42
CA6 P23280 2/20 0.42
DPP4 P27487 2/20 0.42
CA5A P35218 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
CA14 Q9ULX7 2/20 0.42
CA5B Q9Y2D0 2/20 0.42
ESR1 P03372 1/20 0.42
TYR P14679 1/20 0.42
ESR2 Q92731 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4611043 1.00 PKM (0.48) PKMNPSR1HCAR2CA12AKR1B10
SCHEMBL2083461 0.83 CA12 (0.53) CA12CA1CA2DPP4CA7
SCHEMBL9912440 0.80 CA12 (0.59) PKMHCAR2CA12AKR1B10CA1
SCHEMBL31708315 0.80 CA12 (0.59) PKMHCAR2CA12AKR1B10CA1
SCHEMBL13613845 0.78 CYP26B1 (0.62) PKMNPSR1HCAR2CA12AKR1B10
SCHEMBL4612491 0.77 LTB4R (0.51) PKMNPSR1HCAR2CA12AKR1B10
SCHEMBL4612494 0.77 LTB4R (0.51) PKMNPSR1HCAR2CA12AKR1B10
SCHEMBL2083464 0.76 TBXAS1 (0.42) ESR1KDM4EMEN1KMT2APPARG
SCHEMBL2083465 0.76 TBXAS1 (0.42) ESR1KDM4EMEN1KMT2APPARG
SCHEMBL1510128 0.76 HDAC2 (0.58) PKMHCAR2CA12AKR1B10CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781297-B1 NOVEL BIAROMATIC COMPOUNDS THAT ACTIVATE PPAR TYPE RECEPTORS, AND USE THEREOF IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS GALDERMA RES & DEV (FR) 2008-10-15 EP disclosed
EP-1781297-A1 NOVEL BIAROMATIC COMPOUNDS THAT ACTIVATE PPAR TYPE RECEPTORS, AND USE THEREOF IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS Galderma Research & Development, S.N.C. (FR) 2007-05-09 EP disclosed
WO-2006018326-A1 NOVEL BIAROMATIC COMPOUNDS THAT ACTIVATE PPAR TYPE RECEPTORS, AND USE THEREOF IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2006-02-23 WO disclosed