SCHEMBL4617151

SCHEMBL4617151

O=C(O)c1ccc(-c2cccc(CNS(=O)(=O)c3cc(S(=O)(=O)c4ccccc4)ccc3C(F)(F)F)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SFRP1 Q8N474 17/20 0.53
KEAP1 Q14145 1/20 0.49
NFE2L2 Q16236 1/20 0.49
LMNA P02545 1/20 0.46
RAB9A P51151 1/20 0.46
WNT3 P56703 4/20 0.45
CYP19A1 P11511 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4617944 0.93 SFRP1 (0.54) SFRP1KEAP1NFE2L2LMNARAB9A
SCHEMBL4616131 0.92 SFRP1 (0.56) SFRP1WNT3
SCHEMBL4617035 0.91 SFRP1 (0.54) SFRP1LMNARAB9AWNT3
SCHEMBL4618553 0.89 SFRP1 (0.59) SFRP1WNT3
SCHEMBL4618950 0.82 SFRP1 (0.47) SFRP1LMNAWNT3
SCHEMBL4615610 0.81 SFRP1 (0.57) SFRP1WNT3
SCHEMBL4616901 0.81 SFRP1 (0.50) SFRP1LMNAWNT3CYP19A1
SCHEMBL4617361 0.80 POLB (0.58) SFRP1WNT3
SCHEMBL4617471 0.80 SFRP1 (0.54) SFRP1LMNARAB9A
SCHEMBL4617728 0.77 LMNA (0.60) SFRP1LMNARAB9AWNT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP claimed
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof WYETH (US) 2006-12-07 US claimed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO claimed
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP disclosed
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof WYETH (US) 2006-12-07 US disclosed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof SFRP1, SOS1, FZD7 SFRP1 1/4885KEAP1 1841/4885NFE2L2 3293/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.