SCHEMBL4617818

SCHEMBL4617818

CC(C)c1ccc(S(=O)(=O)c2ccccc2)cc1S(=O)(=O)NCCc1cccnc1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SFRP1 Q8N474 2/20 0.58
TBXAS1 P24557 10/20 0.51
NAMPT P43490 3/20 0.47
TDP1 Q9NUW8 1/20 0.46
IDO1 P14902 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4619248 0.92 TBXAS1 (0.53) SFRP1TBXAS1NAMPTIDO1
SCHEMBL4618309 0.89 SFRP1 (0.72) SFRP1
SCHEMBL4617522 0.89 TBXAS1 (0.49) SFRP1TBXAS1NAMPTTDP1
SCHEMBL4618242 0.84 SFRP1 (0.58) SFRP1TBXAS1NAMPTTDP1
SCHEMBL4617566 0.84 SFRP1 (0.62) SFRP1TBXAS1NAMPT
SCHEMBL4616480 0.84 SFRP1 (0.58) SFRP1TBXAS1NAMPTTDP1
SCHEMBL4617716 0.82 TBXAS1 (0.51) SFRP1TBXAS1NAMPT
SCHEMBL4619160 0.82 SFRP1 (0.55) SFRP1TBXAS1NAMPTTDP1
SCHEMBL4617001 0.81 SFRP1 (0.52) SFRP1
SCHEMBL4618668 0.80 ADRB3 (0.48) TBXAS1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP claimed
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof WYETH (US) 2006-12-07 US claimed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO claimed
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP disclosed
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof WYETH (US) 2006-12-07 US disclosed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof SFRP1, SOS1, FZD7 SFRP1 1/4885TBXAS1 2485/4885NAMPT 3852/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.