SCHEMBL4619092

SCHEMBL4619092

CCCc1ccc(S(=O)(=O)c2ccccc2)cc1S(=O)(=O)NCCc1ccccn1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SFRP1 Q8N474 4/20 0.53
RAB9A P51151 1/20 0.52
KDM4E B2RXH2 1/20 0.49
MAPT P10636 1/20 0.49
ADORA3 P0DMS8 3/20 0.47
ADORA2B P29275 3/20 0.47
ADORA1 P30542 3/20 0.47
PRMT5 O14744 1/20 0.44
WDR77 Q9BQA1 1/20 0.44
PKM P14618 1/20 0.44
HTT P42858 1/20 0.43
ATM Q13315 1/20 0.43
LMNA P02545 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6102561 0.94 SFRP1 (0.61) SFRP1RAB9AKDM4EMAPTADORA3
SCHEMBL4617416 0.93 RAB9A (0.49) SFRP1RAB9AKDM4EMAPTADORA3
SCHEMBL4618304 0.86 SFRP1 (0.71) SFRP1RAB9AKDM4EMAPTPRMT5
SCHEMBL4616698 0.84 SFRP1 (0.72) SFRP1HTTALDH1A1
SCHEMBL6101959 0.84 SFRP1 (0.53) SFRP1RAB9AKDM4EMAPTADORA3
SCHEMBL4618264 0.84 TDP1 (0.62) SFRP1PKMHTTLMNATDP1
SCHEMBL4618186 0.84 SFRP1 (0.52) SFRP1RAB9AKDM4EMAPTADORA3
SCHEMBL4615560 0.84 POLB (0.56) SFRP1RAB9AKDM4EMAPTPRMT5
SCHEMBL4616060 0.83 KDM4E (0.71) SFRP1RAB9AKDM4EMAPTPRMT5
SCHEMBL4617001 0.83 SFRP1 (0.52) SFRP1RAB9AKDM4EMAPTADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP claimed
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof WYETH (US) 2006-12-07 US claimed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO claimed
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP disclosed
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof WYETH (US) 2006-12-07 US disclosed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof SFRP1, SOS1, FZD7 SFRP1 1/4885RAB9A 1163/4885KDM4E 3044/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.