SCHEMBL4619429

SCHEMBL4619429

O=C(OCC1(COC(=O)c2ccccc2)COc2ccccc2C1=O)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.41
PRKCA P17252 6/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
TDP1 Q9NUW8 2/20 0.40
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
HIF1A Q16665 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A3 Q01959 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4618060 0.88 GAA (0.47) PRKCA
SCHEMBL4619070 0.85 LMNA (0.43) SMN1; SMN2NPC1RAB9A
SCHEMBL2156979 0.84 PRKCA (0.44) SMN1; SMN2PRKCANPC1RAB9AMAPT
SCHEMBL12395267 0.84 MAPT (0.46) SMN1; SMN2PRKCANPC1RAB9AKMT2A
SCHEMBL4618449 0.79 KMT2A (0.41) SMN1; SMN2NPC1RAB9ATDP1KMT2A
SCHEMBL2156976 0.75 APEX1 (0.44) KMT2AMAPK1
SCHEMBL12395266 0.75 SMN1; SMN2 (0.42) SMN1; SMN2TDP1KMT2AMAPTMAPK1
SCHEMBL4619703 0.74 ALDH1A1 (0.42) SMN1; SMN2PRKCATDP1KMT2AMAPT
SCHEMBL2156506 0.74 FOLH1 (0.41) KMT2AMAPTHIF1A
SCHEMBL2156923 0.71 TSHR (0.39) SMN1; SMN2PRKCAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888555-A2 SUBSTITUTED BENZO-CONDENSED CYCLOHEXANONE DERIVATIVES AND THE USE THEREOF FOR MEDICAMENT PRODUCTION Grünenthal GmbH (DE) 2008-02-20 EP claimed
WO-2006122771-A2 SUBSTITUTED BENZO-CONDENSED CYCLOHEXANONE DERIVATIVES AND THE USE THEREOF FOR MEDICAMENT PRODUCTION Grünenthal GmbH (DE) 2006-11-23 WO claimed
EP-1888555-A2 SUBSTITUTED BENZO-CONDENSED CYCLOHEXANONE DERIVATIVES AND THE USE THEREOF FOR MEDICAMENT PRODUCTION Grünenthal GmbH (DE) 2008-02-20 EP disclosed
WO-2006122771-A2 SUBSTITUTED BENZO-CONDENSED CYCLOHEXANONE DERIVATIVES AND THE USE THEREOF FOR MEDICAMENT PRODUCTION Grünenthal GmbH (DE) 2006-11-23 WO disclosed