SCHEMBL4620127

SCHEMBL4620127

O=C(c1ccc2c(c1)OCO2)N1CCN(CCCOc2cccc3[nH]c4ccccc4c23)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.51
CHRNB2 P17787 1/20 0.51
ACHE P22303 1/20 0.51
CHRNA7 P36544 1/20 0.51
CHRNA4 P43681 1/20 0.51
DRD2 P14416 3/20 0.51
DRD3 P35462 3/20 0.51
HSD17B10 Q99714 2/20 0.47
TSHR P16473 1/20 0.47
GFER P55789 1/20 0.47
ALDH1A1 P00352 7/20 0.47
KDM4E B2RXH2 1/20 0.46
HSD11B1 P28845 1/20 0.45
HPGD P15428 2/20 0.45
PARP1 P09874 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2997062 0.85 ADRB2 (0.59) TSHRSMN1; SMN2
SCHEMBL2992193 0.77 ADRB3 (0.57) HSD11B1LMNA
SCHEMBL18917630 0.76 KMT2A (0.52) HSD17B10ALDH1A1KDM4EHPGDPARP1
SCHEMBL13149543 0.74 ALDH1A1 (0.64) HSD17B10TSHRGFERALDH1A1KDM4E
SCHEMBL2165589 0.73 DRD2 (0.52) DRD2DRD3HSD17B10TSHRGFER
SCHEMBL2998745 0.72 ADRB2 (0.53) ALDH1A1KDM4EHPGDCYP1A2CYP3A4
SCHEMBL2998748 0.72 ADRB2 (0.53) ALDH1A1KDM4EHPGDCYP1A2CYP3A4
SCHEMBL18029394 0.71 ALDH1A1 (0.68) DRD2DRD3HSD17B10TSHRGFER
SCHEMBL9412168 0.71 ALDH1A1 (0.63) HSD17B10TSHRGFERALDH1A1KDM4E
SCHEMBL2997254 0.70 MEN1 (0.64) TSHRKDM4ESMN1; SMN2HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP disclosed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO disclosed