SCHEMBL4623518

SCHEMBL4623518

CC(C)(C)c1cccc(OCc2ccc(-c3ccc(C(=O)N([C@@H](CCC(N)=O)C(=O)O)C(C)(C)Cc4ccccc4)cc3)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 3/20 0.43
NR4A2 P43354 3/20 0.42
NR4A1 P22736 1/20 0.42
NR4A3 Q92570 1/20 0.42
PTGES O14684 2/20 0.41
ALOX5 P09917 2/20 0.41
LTC4S Q16873 1/20 0.41
SPHK2 Q9NRA0 3/20 0.40
KMT2A Q03164 1/20 0.38
SMPD1 P17405 1/20 0.38
SPHK1 Q9NYA1 1/20 0.38
PKM P14618 1/20 0.37
CACNA1B Q00975 1/20 0.37
MAOB P27338 1/20 0.37
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4622870 0.94 PSEN1 (0.38) BCL2NR4A2NR4A1NR4A3PTGES
SCHEMBL2247850 0.91 PTGES (0.43) BCL2NR4A2NR4A1NR4A3PTGES
SCHEMBL2244683 0.91 SPHK2 (0.43) PTGESALOX5LTC4SSPHK2KMT2A
SCHEMBL2249360 0.90 BCL2 (0.43) BCL2NR4A2NR4A1NR4A3PTGES
SCHEMBL4374329 0.89 PSEN1 (0.44) BCL2NR4A2PTGESALOX5KMT2A
SCHEMBL2250531 0.86 HSD17B2 (0.43) PTGESALOX5LTC4SPKMMAOB
SCHEMBL2249759 0.85 RXRA (0.47) PTGESALOX5LTC4SRXRARXRB
SCHEMBL2243828 0.84 EPOR (0.38) BCL2NR4A2NR4A1NR4A3PTGES
SCHEMBL2245867 0.83 MMP2 (0.40) PTGESALOX5
SCHEMBL2244933 0.83 HSD17B2 (0.51) PTGESALOX5KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902014-A2 GLUTAMATE AGGRECANASE INHIBITORS Wyeth (US) 2008-03-26 EP disclosed
WO-2007008994-A2 GLUTAMATE AGGRECANASE INHIBITORS WYETH (US) 2007-01-18 WO disclosed