SCHEMBL4623908

SCHEMBL4623908

CSc1ccc2c(c1)c1c(n2S(=O)(=O)c2ccc(C)cc2)CC[CH]C1

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 18/20 0.66
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4623910 0.82 HTR6 (0.64) HTR6PTGS1PTGS2MAPT
SCHEMBL833490 0.79 HTR6 (1.00) HTR6
SCHEMBL12868529 0.70 HTR6 (0.78) HTR6
SCHEMBL835912 0.69 HTR6 (1.00) HTR6
SCHEMBL8036424 0.68 HTR6 (0.68) HTR6PTGS1PTGS2MAPT
SCHEMBL12868160 0.67 HTR6 (0.64) HTR6PTGS1PTGS2MAPT
SCHEMBL5325197 0.67 HTR6 (0.52) HTR6MAPT
SCHEMBL5325199 0.66 HTR6 (0.51) HTR6MAPT
SCHEMBL21114803 0.66 HTR6 (0.63) HTR6
SCHEMBL24219916 0.65 PKM (0.50) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948166-A1 CARBAZOLE DERIVATIVES AS FUNCTIONAL 5-HT6 LIGANDS Suven Life Sciences Limited (IN) 2008-07-30 EP disclosed
WO-2007046111-A1 CARBAZOLE DERIVATIVES AS FUNCTIONAL 5-HT6 LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2007-04-26 WO disclosed