SCHEMBL462541

SCHEMBL462541

CC(C(=O)O)c1ccc(I)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.61
PTGS1 P23219 8/20 0.57
AKR1C3 P42330 8/20 0.57
AKR1C2 P52895 7/20 0.57
CYP2C9 P11712 4/20 0.57
LMNA P02545 3/20 0.57
CXCR1 P25024 2/20 0.57
CXCR2 P25025 2/20 0.57
SLC22A6 Q4U2R8 2/20 0.57
TSHR P16473 2/20 0.57
ALB P02768 1/20 0.57
ESR1 P03372 1/20 0.57
ALOX5 P09917 1/20 0.57
RARB P10826 1/20 0.57
ADRB3 P13945 1/20 0.57
NFKB1 P19838 1/20 0.57
HTR2A P28223 1/20 0.57
NR1I3 Q14994 1/20 0.57
CXCL8 P10145 1/20 0.57
BLM P54132 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11483097 0.98 PTGS2 (0.59) PTGS2PTGS1AKR1C3AKR1C2CYP2C9
SCHEMBL59197 0.88 PTGS2 (0.74) PTGS2PTGS1AKR1C3AKR1C2CYP2C9
SCHEMBL11724969 0.85 AKR1C3 (0.63) PTGS2PTGS1AKR1C3AKR1C2CYP2C9
SCHEMBL27536644 0.84 ACACB (0.46) PTGS2PTGS1AKR1C3AKR1C2CYP2C9
SCHEMBL6551674 0.81 PTGS2 (0.65) PTGS2PTGS1AKR1C3AKR1C2CYP2C9
SCHEMBL917093 0.81 PTGS2 (0.87) PTGS2PTGS1AKR1C3AKR1C2CYP2C9
SCHEMBL4651605 0.81 PTGS2 (0.65) PTGS2PTGS1AKR1C3AKR1C2CYP2C9
SCHEMBL459261 0.80 EPHX1 (0.58) PTGS2PTGS1AKR1C3AKR1C2CYP2C9
SCHEMBL29318759 0.80 ACACB (0.43) PTGS2PTGS1AKR1C3AKR1C2CYP2C9
SCHEMBL10333915 0.79 PTGS1 (0.59) PTGS2PTGS1AKR1C3AKR1C2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 113 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-5140028-A None JP disclosed
JP-5140028-A None JP disclosed
CN-118955244-A Method for preparing primary alcohol by homogeneously catalyzing and reducing carboxylic acid derivative by using N-heterocyclic carbene copper complex 延安大学 2024-11-15 CN disclosed
CN-118076367-A GLP-1 receptor agonists with improved pharmacological and drug delivery properties 达比克斯有限责任公司 2024-05-24 CN disclosed
CN-114292226-B Compound with hydroxamic acid structure and preparation method and application thereof 沈阳药科大学 2023-04-18 CN disclosed
CN-112479921-B Compound with PPAR delta agonist activity, pharmaceutical composition and medical application 中国药科大学 2022-12-06 CN disclosed
CN-114292226-A Compound with hydroxamic acid structure and preparation method and application thereof 沈阳药科大学 2022-04-08 CN disclosed
CN-109970542-B Application of quebrachitol in copper-catalyzed aryl halide hydrolysis reaction 沈阳药科大学 2021-06-11 CN disclosed
CN-112479921-A Compound with PPAR delta agonist activity, pharmaceutical composition and medical application 中国药科大学 2021-03-12 CN disclosed
CN-111704912-A Novel preparation method of 3-alkenyl benzyne liquid crystal compound 烟台丰蓬液晶材料有限公司 2020-09-25 CN disclosed
US-6359135-B1 Compounds having activity as inhibitors of cytochrome P450RAI ALLERGAN SALES, INC. 2002-03-19 US disclosed
WO-2002018361-A2 COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF CYTOCHROME P450RAI ALLERGAN, INC. (US) 2002-03-07 WO disclosed
US-6313107-B1 ADMINISTERING TO MAMMAL TO TREAT DISEASES RESPONSIVE TO TREATMENT BY RETINOIDS ALLERGAN SALES, INC. 2001-11-06 US disclosed
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed
US-6291677-B1 FOR TREATING SKIN-RELATED DISEASES, INCLUDING, ACTINIC KERATOSES, ARSENIC KERATOSES, INFLAMMATORY AND NON-INFLAMMATORY ACNE, PSORIASIS, ICHTHYOSES AND KERATINIZATION AND HYPERPROLIFERATIVE DISORDERS OF SKIN ALLERGAN SALES, INC. 2001-09-18 US disclosed
US-6252090-B1 Compounds having activity as inhibitors of cytochrome P450RAI ALLERGAN SALES, INC. 2001-06-26 US disclosed
JP-H05140028-A PRODUCTION OF 2-(4-IODOPHENYL)-PROPIONIC ACID AND ITS ESTER NAGASE SANGYO KK 1993-06-08 JP disclosed
JP-H05140028-A PRODUCTION OF 2-(4-IODOPHENYL)-PROPIONIC ACID AND ITS ESTER NAGASE SANGYO KK 1993-06-08 JP disclosed
US-4252719-A REMOVAL OF A TERTIARY HYDROGEN FROM A 5-A-STEROID BY CHLORINATING THE STEROID BEING FIRST ESTERIFIED BY AN IODOARYL-CONTAINING ESTERIFICATION AGENT RESEARCH CORPORATION (US) 1981-02-24 US disclosed
US-4230719-A Novel 2-[4-(3-methyl-2-thienyl)phenyl]propionic acid and pharmaceutically acceptable salt thereof and method for treating symptoms of inflammation and pain TOYAMA CHEMICAL CO., LTD. (JP) 1980-10-28 US disclosed