SCHEMBL4625979

SCHEMBL4625979

CN(C)C1CCN(S(=O)(=O)c2cccc3c(Nc4cccc5c4CCO5)c(C(N)=O)cnc23)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 4/20 0.54
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35
MTNR1B P49286 1/20 0.35
CSF1R P07333 4/20 0.34
KCNH2 Q12809 1/20 0.34
JAK2 O60674 1/20 0.34
JAK3 P52333 1/20 0.34
GAA P10253 1/20 0.34
ALDH1A1 P00352 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4628806 0.88 PDE4B (0.57) PDE4BMTNR1BCSF1RGAAALDH1A1
SCHEMBL4627538 0.88 PDE4B (0.54) PDE4BMTNR1BCSF1RJAK2JAK3
SCHEMBL4627674 0.87 PDE4B (0.56) PDE4BALOX5APFEN1MTNR1BCSF1R
SCHEMBL4625977 0.85 PDE4B (0.71) PDE4BCSF1RKCNH2
Hydrochloric Acid SCHEMBL4628811 0.85 PDE4B (0.70) PDE4BCSF1RKCNH2
SCHEMBL4949173 0.83 PDE4B (0.69) PDE4BMTNR1BCSF1RJAK2JAK3
SCHEMBL4627082 0.82 PDE4B (0.51) PDE4BMTNR1BCSF1RKCNH2ALDH1A1
SCHEMBL4628322 0.80 PDE4B (0.57) PDE4BMTNR1BCSF1RKCNH2GAA
SCHEMBL4626847 0.80 PDE4B (0.56) PDE4BMTNR1BCSF1RKCNH2
SCHEMBL5404792 0.79 PDE4B (0.51) PDE4BMTNR1BCSF1RPDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673086-B1 4-AMINOQUINOLINE-3-CARBOXAMIDE DERIVATIVES AS PDE4 INHIBITORS GLAXO GROUP LTD (GB) 2008-01-23 EP claimed