SCHEMBL4627675

SCHEMBL4627675

NC(=O)c1cnc2ccc(SSc3ccc4ncc(C(N)=O)c(Cl)c4c3)cc2c1Cl

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.48
PDE4B Q07343 7/20 0.43
LMNA P02545 1/20 0.41
CSF1R P07333 5/20 0.38
ATM Q13315 2/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
MTOR P42345 1/20 0.38
PIK3CG P48736 1/20 0.38
PRKDC P78527 1/20 0.38
ATR Q13535 1/20 0.38
NNMT P40261 2/20 0.38
KDM4E B2RXH2 1/20 0.37
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4628822 0.85 SLC2A1 (0.65) SLC2A1PDE4BLMNACSF1RATM
SCHEMBL9875438 0.83 LMNA (0.56) SLC2A1PDE4BLMNACSF1RATM
SCHEMBL2479384 0.81 LMNA (0.42) SLC2A1PDE4BLMNACSF1RATM
SCHEMBL3866828 0.81 CSF1R (0.46) SLC2A1PDE4BLMNACSF1R
SCHEMBL2725311 0.81 HTT (0.49) SLC2A1PDE4BLMNACSF1RKDM4E
SCHEMBL5929785 0.78 NNMT (0.46) SLC2A1LMNACSF1RATMNNMT
SCHEMBL3273151 0.77 KDM4E (0.64) PDE4BLMNACSF1RKDM4E
SCHEMBL4657732 0.77 PDE4B (0.49) PDE4B
SCHEMBL2706557 0.76 KMT2A (0.47) SLC2A1PDE4BLMNACSF1RATM
SCHEMBL18318006 0.75 CSF1R (0.49) SLC2A1CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080096884-A1 4-Aminoquinoline-3-Carboxamide Derivatives as Pde4 Inhibitors GLAXO GROUP LIMITED (GB) 2008-04-24 US disclosed
US-20080096884-A1 4-Aminoquinoline-3-Carboxamide Derivatives as Pde4 Inhibitors GLAXO GROUP LIMITED (GB) 2008-04-24 US disclosed
US-20080096884-A1 4-Aminoquinoline-3-Carboxamide Derivatives as Pde4 Inhibitors GLAXO GROUP LIMITED (GB) 2008-04-24 US disclosed
EP-1673086-B1 4-AMINOQUINOLINE-3-CARBOXAMIDE DERIVATIVES AS PDE4 INHIBITORS GLAXO GROUP LTD (GB) 2008-01-23 EP disclosed
EP-1673086-B1 4-AMINOQUINOLINE-3-CARBOXAMIDE DERIVATIVES AS PDE4 INHIBITORS GLAXO GROUP LTD (GB) 2008-01-23 EP disclosed
EP-1673086-A1 4-AMINOQUINOLINE-3-CARBOXAMIDE DERIVATIVES AS PDE4 INHIBITORS GLAXO GROUP LIMITED (GB) 2006-06-28 EP disclosed
WO-2005030212-A1 4-AMINOQUINOLINE-3-CARBOXAMIDE DERIVATIVES AS PDE4 INHIBITORS GLAXO GROUP LIMITED (GB) 2005-04-07 WO disclosed
WO-2005030212-A1 4-AMINOQUINOLINE-3-CARBOXAMIDE DERIVATIVES AS PDE4 INHIBITORS GLAXO GROUP LIMITED (GB) 2005-04-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080096884-A1 4-Aminoquinoline-3-Carboxamide Derivatives as Pde4 Inhibitors PDE4A, PDE4B, PDE3B SLC2A1 4263/4885PDE4B 2/4885LMNA 3636/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.