SCHEMBL4627985

SCHEMBL4627985

CCOC(=O)O[C@@H]1CCCN1C1CCNCC1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.39
ALDH1A1 P00352 4/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
THRB P10828 1/20 0.35
ATM Q13315 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
GAA P10253 2/20 0.34
TP53 P04637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CHRM1 P11229 1/20 0.33
TPSAB1 Q15661 2/20 0.32
TPSD1 Q9BZJ3 2/20 0.32
TPSG1 Q9NRR2 2/20 0.32
MAPK1 P28482 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4604392 0.84 SLC6A2 (0.33) SLC6A2SLC6A4SLC6A3TPSAB1TPSD1
SCHEMBL4628886 0.83 POLB (0.34) POLBALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL4720288 0.83 POLB (0.34) POLBALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL1207252 0.77 FKBP1A (0.42) POLBALDH1A1KDM4EMAPK1
SCHEMBL4629748 0.75 POLB (0.37) POLBALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL4718582 0.75 TP53 (0.34) POLBALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL4719694 0.75 POLB (0.37) POLBALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL5176485 0.73 FKBP1A (0.47) POLBALDH1A1KDM4EMAPK1
SCHEMBL1461712 0.72 ALDH1A1 (0.44) ALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL4717467 0.68 ALDH1A1 (0.36) ALDH1A1SLC6A2SLC6A4SLC6A3GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917256-A2 SELECTED CGRP ANTAGONISTS, METHODS FOR THE PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS Boehringer Ingelheim International GmbH (DE) 2008-05-07 EP disclosed
WO-2007020261-A2 SELECTED CGRP ANTAGONISTS, METHODS FOR THE PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-02-22 WO disclosed