SCHEMBL4628562

SCHEMBL4628562

Oc1ccc(-c2ccccc2)c(C(F)(F)F)c1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.43
ALOX5 P09917 2/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
BCL2L1 Q07817 1/20 0.42
HSD17B10 Q99714 1/20 0.42
GYS1 P13807 1/20 0.39
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
KIF11 P52732 1/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
CNR1 P21554 1/20 0.36
NR2F2 P24468 1/20 0.36
CNR2 P34972 1/20 0.36
KMT2A Q03164 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36
ESR2 Q92731 3/20 0.35
CYP17A1 P05093 1/20 0.35
CYP11B1 P15538 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28431087 0.83 GYS1 (0.47) BACE1ALOX5ALDH1A1HPGDBCL2L1
SCHEMBL27727564 0.80 BACE1 (0.42) BACE1ALOX5ALDH1A1HPGDBCL2L1
SCHEMBL1513817 0.78 BACE1 (0.52) BACE1ALOX5ALDH1A1HPGDBCL2L1
SCHEMBL27967295 0.77 ALDH1A1 (0.41) BACE1ALOX5ALDH1A1HPGDBCL2L1
SCHEMBL27587157 0.77 PTPN1 (0.44) HPGDLMNAMEN1MAPTKMT2A
SCHEMBL5132773 0.77 ALDH1A1 (0.56) BACE1ALOX5ALDH1A1HPGDBCL2L1
SCHEMBL321984 0.76 BACE1 (0.42) BACE1ALOX5ALDH1A1HPGDBCL2L1
SCHEMBL29351964 0.76 BACE1 (0.50) BACE1ALOX5ALDH1A1HPGDBCL2L1
SCHEMBL27692000 0.76 BACE1 (0.50) BACE1ALOX5ALDH1A1HPGDBCL2L1
SCHEMBL2654207 0.76 BACE1 (0.38) BACE1ALOX5ALDH1A1HPGDBCL2L1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917240-A1 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2008-05-07 EP disclosed
WO-2007024922-A1 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2007-03-01 WO disclosed