SCHEMBL4629548

SCHEMBL4629548

CNc1cc(C)c(OCCCC2CNCCN2c2cccc3sccc23)c(OC)c1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.34
HTR1A P08908 7/20 0.34
HTR2A P28223 7/20 0.34
HTR2C P28335 1/20 0.33
ADRA1A P35348 1/20 0.33
HRH1 P35367 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4629376 0.89 DRD2 (0.33) DRD2HTR1AHTR2A
Hydrochloric Acid SCHEMBL4631048 0.83 HTR1A (0.33) DRD2HTR1AHTR2AHTR2CADRA1A
Hydrochloric Acid SCHEMBL4630605 0.83 HTR1A (0.33) DRD2HTR1AHTR2AHTR2CADRA1A
SCHEMBL4630236 0.79 DRD2 (0.45) DRD2HTR1AHTR2AHTR2CADRA1A
SCHEMBL294686 0.78 HTR2A (0.53) DRD2HTR1AHTR2AHTR2CADRA1A
Hydrochloric Acid SCHEMBL294382 0.78 HTR2A (0.53) DRD2HTR1AHTR2AHTR2CADRA1A
Hydrochloric Acid SCHEMBL4630464 0.74 DRD2 (0.33) DRD2HTR1AHTR2AHTR2CADRA1A
Hydrochloric Acid SCHEMBL5508259 0.71 DRD2 (0.42) DRD2
SCHEMBL5504510 0.70 HTR1A (0.38) DRD2HTR1AHTR2AHTR2CADRA1A
SCHEMBL20915103 0.70 DRD2 (0.46) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed