SCHEMBL4629945

SCHEMBL4629945

CCCc1cc([O])ccc1-c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.39
PPARA Q07869 1/20 0.38
DPP4 P27487 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
KMT2A Q03164 1/20 0.36
CSNK2A1 P68400 2/20 0.35
FOLH1 Q04609 1/20 0.35
PTGER1 P34995 1/20 0.35
PTGER4 P35408 1/20 0.35
PTGER3 P43115 1/20 0.35
PTGER2 P43116 1/20 0.35
PTGS1 P23219 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4630596 0.90 PSMB5 (0.40) PPARA
SCHEMBL4629849 0.88 GPR84 (0.42) PPARA
SCHEMBL4629941 0.87 DPP4 (0.41) MAPTDPP4ADORA3ADORA2AADORA1
SCHEMBL4630629 0.87 BID (0.43) PPARA
SCHEMBL10798309 0.81 SMN1; SMN2 (0.40) MAPTPPARADPP4ADORA3ADORA2A
SCHEMBL28312672 0.80 CA12 (0.42) MAPTDPP4ADORA3ADORA2AADORA1
SCHEMBL29795424 0.79 DPP4 (0.41) MAPTDPP4ADORA3ADORA2AADORA1
SCHEMBL6517710 0.79 PTGDR2 (0.40) MAPTPPARADPP4ADORA3ADORA2A
SCHEMBL28600186 0.79 ALOX5 (0.55) ESR2PTPN1PTPN11BACE1ALOX5
SCHEMBL12505671 0.78 PPARG (0.50) MAPTFOLH1PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed