SCHEMBL4629985

SCHEMBL4629985

CCCC[CH]c1ccn[nH]1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP19A1 P11511 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
KMT2A Q03164 1/20 0.36
COMT P21964 4/20 0.36
CTH P32929 1/20 0.34
SCN4A P35499 2/20 0.31
PDPK1 O15530 1/20 0.31
TLK2 Q86UE8 2/20 0.31
USP2 O75604 1/20 0.31
LMNA P02545 1/20 0.31
HRH2 P25021 1/20 0.31
HPGDS O60760 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4629924 0.88
SCHEMBL15106949 0.69
SCHEMBL6687128 0.67 GAA (0.46) KMT2APDPK1TLK2LMNA
SCHEMBL8200303 0.65 MAPT (0.44) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL181391 0.65 CYP1A2 (0.40) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL6320373 0.65 ALDH1A1 (0.39) KMT2ALMNA
SCHEMBL658444 0.64 USP2 (0.55) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL19361929 0.63
SCHEMBL543822 0.63
SCHEMBL25530345 0.63 USP2 (0.53) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed