SCHEMBL463000

SCHEMBL463000

Cn1c(-c2cncc(F)c2)nc2c(F)c(F)ccc21

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 6/20 0.41
CYP11B1 P15538 4/20 0.41
CYP19A1 P11511 1/20 0.40
ADRA2B P18089 1/20 0.40
TLR7 Q9NYK1 12/20 0.40
GRIN1 Q05586 2/20 0.38
GRIN2B Q13224 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12505500 0.84 PDE2A (0.50) CYP11B2CYP11B1TLR7
SCHEMBL462661 0.83 CYP11B2 (0.46) CYP11B2CYP11B1TLR7
SCHEMBL17896720 0.80 CYP11B1 (0.43) CYP11B2CYP11B1CYP19A1ADRA2BTLR7
SCHEMBL10176205 0.78 CYP11B2 (0.56) CYP11B2CYP11B1CYP19A1ADRA2BTLR7
SCHEMBL17896718 0.77 CYP11B2 (0.56) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL17896599 0.75 CYP11B2 (0.63) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL10175581 0.74 CYP11B2 (0.71) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL17896665 0.74 KDM4E (0.52) CYP11B2CYP11B1CYP19A1ADRA2BTLR7
SCHEMBL17896619 0.74 NPC1 (0.51) CYP11B2CYP11B1CYP19A1ADRA2BTLR7
SCHEMBL17896687 0.74 CYP11B1 (0.55) CYP11B2CYP11B1CYP19A1ADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595482-A1 ALDOSTERONE SYNTHASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-29 EP disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed