SCHEMBL10176205

SCHEMBL10176205

Cn1c(-c2cncc(F)c2)nc2ccc(F)c(F)c21

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 14/20 0.56
CYP11B1 P15538 12/20 0.46
CYP19A1 P11511 2/20 0.46
ADRA2B P18089 2/20 0.46
ADRB1 P08588 1/20 0.37
ADRA2A P08913 1/20 0.37
ADRA2C P18825 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
GRIN1 Q05586 2/20 0.35
GRIN2B Q13224 2/20 0.35
TLR7 Q9NYK1 2/20 0.35
PIK3CG P48736 1/20 0.34
PIM1 P11309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175459 0.89 CYP11B2 (0.56) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
SCHEMBL17896705 0.86 CYP11B2 (0.54) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
SCHEMBL17897057 0.84 CYP11B2 (0.52) CYP11B2CYP11B1
SCHEMBL17896707 0.84 CYP11B2 (0.52) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
SCHEMBL10175455 0.83 CYP11B2 (0.51) CYP11B2CYP11B1TLR7PIK3CG
SCHEMBL10176201 0.82 CYP11B2 (0.64) CYP11B2CYP11B1CYP19A1ADRA2BADRB1
SCHEMBL17896770 0.81 CYP11B2 (0.40) CYP11B2CYP11B1CYP19A1ADRA2BTLR7
SCHEMBL10175447 0.81 CYP11B2 (0.60) CYP11B2CYP11B1
SCHEMBL17896600 0.80 CYP11B2 (0.45) CYP11B2CYP11B1CYP19A1ADRA2BTLR7
SCHEMBL463000 0.78 CYP11B2 (0.41) CYP11B2CYP11B1CYP19A1ADRA2BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed