SCHEMBL4630547

SCHEMBL4630547

O=C(CO)C1CCCCN1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 2/20 0.43
NOS2 P35228 2/20 0.39
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
PRCP P42785 1/20 0.38
DPP4 P27487 4/20 0.37
DPP8 Q6V1X1 2/20 0.36
DPP9 Q86TI2 2/20 0.36
HTR2B P41595 2/20 0.36
HTR2C P28335 1/20 0.36
FAP Q12884 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
CYP2D6 P10635 2/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15307927 1.00 FDPS (0.43) FDPSNOS2NOS3NOS1PRCP
SCHEMBL17929297 1.00 FDPS (0.43) FDPSNOS2NOS3NOS1PRCP
SCHEMBL9040662 0.98 FDPS (0.42) FDPSNOS2NOS3NOS1PRCP
SCHEMBL4630954 0.93
SCHEMBL17929302 0.93
SCHEMBL887204 0.93
Hydrochloric Acid SCHEMBL10834143 0.91 NOS2 (0.43) NOS2NOS3NOS1PRCPDPP4
Hydrochloric Acid SCHEMBL10834147 0.91 NOS2 (0.43) NOS2NOS3NOS1PRCPDPP4
SCHEMBL31463812 0.83 FDPS (0.37) FDPSNOS2NOS3NOS1PRCP
SCHEMBL11872839 0.81 PRCP (0.40) FDPSNOS2NOS3NOS1PRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160297792-A1 PIPERIDINE OR PIPERAZINE LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG MERCK SHARP & DOHME CORP. (US) 2016-10-13 US disclosed
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160297792-A1 PIPERIDINE OR PIPERAZINE LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG CYP3A5, CYP3A43, CYP3A7 FDPS 763/4885NOS2 301/4885NOS3 444/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.