SCHEMBL4630987

SCHEMBL4630987

COCCCCC(=O)C1CNCCN1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
REN P00797 16/20 0.38
TSHR P16473 1/20 0.31
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2701364 0.95 REN (0.39) ALDH1A1RENTSHR
SCHEMBL4630110 0.89 REN (0.36) REN
SCHEMBL28874795 0.82 PRCP (0.41) ALDH1A1TSHR
SCHEMBL4630457 0.81 PRCP (0.44) ALDH1A1TSHR
SCHEMBL4630350 0.80 PRCP (0.39) ALDH1A1
SCHEMBL5543593 0.79
SCHEMBL5537138 0.78
SCHEMBL4630213 0.76 HSD17B10 (0.35)
SCHEMBL4630220 0.74 SLC6A1 (0.31)
SCHEMBL27468849 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed