SCHEMBL4631003

SCHEMBL4631003

Cc1sc(NCC2CC2)nc1-c1ccccc1C#N

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
ACHE P22303 6/20 0.39
NPY5R Q15761 4/20 0.38
CRHR1 P34998 3/20 0.37
CHUK O15111 1/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
NISCH Q9Y2I1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2581646 0.78 ALDH1A1 (0.52) ALDH1A1ACHEMAOAMAOB
SCHEMBL2586747 0.69 ALDH1A1 (0.53) ALDH1A1ACHEMAOAMAOBCYP1A2
SCHEMBL6670189 0.67 KDM4E (0.54) CHUKHSD17B10
SCHEMBL12609243 0.64 CRHR1 (0.49) ALDH1A1ACHECRHR1HSD17B10
SCHEMBL22630233 0.63 ACP1 (0.34) CHUKCYP1A2CYP3A4HSD17B10TDP1
SCHEMBL2638722 0.63 CRHR1 (0.48) ALDH1A1CRHR1HSD17B10
SCHEMBL29691084 0.62 TSHR (0.41) ALDH1A1CYP1A2NISCH
SCHEMBL22616537 0.61 F2R (0.33) CYP1A2CYP3A4HSD17B10TDP1
SCHEMBL5414519 0.60 JAK2 (0.54)
SCHEMBL8791236 0.59 ALDH1A1 (0.46) ALDH1A1HSD17B10NISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924561-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS Eli Lilly & Company (US) 2008-05-28 EP disclosed
WO-2007028083-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2007-03-08 WO disclosed