SCHEMBL4631344

SCHEMBL4631344

Cc1ccccc1NCC(=O)Nc1ccc(-c2ccncc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.67
PORCN Q9H237 1/20 0.49
ALDH1A1 P00352 4/20 0.49
LMNA P02545 2/20 0.49
PKM P14618 1/20 0.49
ADRA2C P18825 1/20 0.48
NAMPT P43490 2/20 0.47
ROCK2 O75116 4/20 0.47
ROCK1 Q13464 4/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
HPGD P15428 1/20 0.46
MAPT P10636 2/20 0.46
OPRK1 P41145 1/20 0.46
TYK2 P29597 1/20 0.46
GRK2 P25098 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4630900 0.85 NOTUM (0.48) NOTUMPORCNALDH1A1ROCK2ROCK1
SCHEMBL6716890 0.83 NOTUM (0.72) NOTUMALDH1A1LMNAMEN1KMT2A
SCHEMBL4630981 0.83 NOTUM (0.46) NOTUMPORCNADRA2CNAMPTROCK2
SCHEMBL4518077 0.82 PORCN (0.64) PORCNALDH1A1LMNAROCK2ROCK1
SCHEMBL4630930 0.81 PORCN (0.46) NOTUMPORCNALDH1A1LMNAROCK2
SCHEMBL4630248 0.81 PORCN (0.46) NOTUMPORCNALDH1A1LMNAROCK2
Hydrochloric Acid SCHEMBL4522424 0.81 PORCN (0.63) PORCNALDH1A1LMNAROCK2ROCK1
SCHEMBL20941790 0.77 NOTUM (0.57) NOTUMALDH1A1LMNAPKMMEN1
SCHEMBL6715566 0.77 NOTUM (0.60) NOTUMALDH1A1LMNAMEN1KMT2A
Trifluoroacetic Acid SCHEMBL4535893 0.75 PORCN (0.57) PORCNALDH1A1LMNAROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1922306-A2 AMIDE DERIVATIVES AS ROCK INHIBITORS Astellas Pharma Inc. (JP) 2008-05-21 EP disclosed
WO-2007026920-A2 AMIDE DERIVATIVES AS ROCK INHIBITORS ASTELLAS PHARMA INC. (JP) 2007-03-08 WO disclosed