SCHEMBL4630248

SCHEMBL4630248

O=C(CNc1ccccc1CCO)Nc1ccc(-c2ccncc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PORCN Q9H237 1/20 0.46
ROCK2 O75116 6/20 0.46
ROCK1 Q13464 6/20 0.46
NOTUM Q6P988 1/20 0.44
GRK2 P25098 1/20 0.44
LMNA P02545 2/20 0.42
ALDH1A1 P00352 4/20 0.42
TDP1 Q9NUW8 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
POLB P06746 1/20 0.40
STAT3 P40763 1/20 0.40
NPY5R Q15761 1/20 0.40
NPC1 O15118 1/20 0.40
MITF O75030 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4631344 0.81 NOTUM (0.67) PORCNROCK2ROCK1NOTUMGRK2
SCHEMBL4630930 0.81 PORCN (0.46) PORCNROCK2ROCK1NOTUMLMNA
SCHEMBL4630900 0.79 NOTUM (0.48) PORCNROCK2ROCK1NOTUMALDH1A1
SCHEMBL4518077 0.79 PORCN (0.64) PORCNROCK2ROCK1GRK2LMNA
Hydrochloric Acid SCHEMBL4522424 0.78 PORCN (0.63) PORCNROCK2ROCK1GRK2LMNA
SCHEMBL4630981 0.77 NOTUM (0.46) PORCNROCK2ROCK1NOTUM
SCHEMBL4520975 0.73 ROCK2 (0.53) ROCK2ROCK1LMNAALDH1A1MEN1
Trifluoroacetic Acid SCHEMBL4535893 0.72 PORCN (0.57) PORCNROCK2ROCK1GRK2LMNA
SCHEMBL11178746 0.72 AAK1 (0.55) ROCK2ROCK1ALDH1A1HTTSMN1; SMN2
SCHEMBL4524018 0.71 LMNA (0.55) ROCK2ROCK1NOTUMLMNANPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1922306-A2 AMIDE DERIVATIVES AS ROCK INHIBITORS Astellas Pharma Inc. (JP) 2008-05-21 EP disclosed
WO-2007026920-A2 AMIDE DERIVATIVES AS ROCK INHIBITORS ASTELLAS PHARMA INC. (JP) 2007-03-08 WO disclosed