SCHEMBL4632242

SCHEMBL4632242

CN(C)C(=O)c1cc([N+](=O)[O-])c(N)c([N+](=O)[O-])c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.53
HTT P42858 1/20 0.53
ALDH1A1 P00352 4/20 0.49
LMNA P02545 3/20 0.49
MEN1 O00255 1/20 0.46
HPGD P15428 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HCAR3 P49019 1/20 0.45
ERN1 O75460 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.41
HKDC1 Q2TB90 1/20 0.41
SLC6A4 P31645 1/20 0.41
TSHR P16473 1/20 0.41
CYP3A4 P08684 1/20 0.41
CASP6 P55212 1/20 0.41
PARP1 P09874 1/20 0.40
ATM Q13315 1/20 0.40
GSTP1 P09211 1/20 0.39
GSTM2 P28161 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4633313 0.92 KMT2A (0.49) KMT2AHTTALDH1A1LMNAMEN1
SCHEMBL29447926 0.90 KMT2A (0.47) KMT2AHTTALDH1A1LMNAMEN1
SCHEMBL25253595 0.90 KMT2A (0.47) KMT2AHTTALDH1A1LMNAMEN1
SCHEMBL25298464 0.90 ALDH1A1 (0.51) KMT2AHTTALDH1A1LMNAMEN1
SCHEMBL29809012 0.90 ALDH1A1 (0.51) KMT2AHTTALDH1A1LMNAMEN1
SCHEMBL22115119 0.81 LMNA (0.66) KMT2AHTTALDH1A1LMNAMEN1
SCHEMBL3106666 0.77 SMN1; SMN2 (0.59) HTTALDH1A1LMNAL3MBTL1TSHR
SCHEMBL865237 0.77 LMNA (0.65) ALDH1A1LMNAHCAR3TSHRCYP3A4
SCHEMBL11350169 0.77 KMT2A (0.68) KMT2AHTTALDH1A1LMNAMEN1
SCHEMBL5914014 0.76 TSHR (0.68) KMT2AHTTALDH1A1LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1926714-A1 ISOTOPICALLY SUBSTITUTED BENZIMIDAZOLE DERIVATIVES Nycomed GmbH (DE) 2008-06-04 EP disclosed
WO-2008017466-A1 PHARMACEUTICALLY ACTIVE TETRAHYDROISOQUINOLINE-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-02-14 WO disclosed
WO-2007023135-A1 ISOTOPICALLY SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2007-03-01 WO disclosed