SCHEMBL4633871

SCHEMBL4633871

N#Cc1ccc(OCCOc2c(C(=O)O)sc3ccccc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 1/20 0.56
PTPN2 P17706 1/20 0.46
PTPN1 P18031 1/20 0.46
MAPT P10636 3/20 0.46
ALDH1A1 P00352 2/20 0.46
MMP2 P08253 2/20 0.45
PRSS12 P56730 1/20 0.44
MCL1 Q07820 3/20 0.44
BCL2 P10415 2/20 0.44
BCL2L1 Q07817 2/20 0.44
BAD Q92934 2/20 0.44
MMP3 P08254 3/20 0.43
EDNRA P25101 1/20 0.42
RXFP1 Q9HBX9 2/20 0.41
LMNA P02545 1/20 0.41
KCNA5 P22460 2/20 0.41
PKM P14618 2/20 0.41
MAOB P27338 1/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4633866 0.88 CXCR2 (0.67) CXCR2PTPN2PTPN1MAPTALDH1A1
SCHEMBL4633951 0.85 KDM4E (0.53) PTPN2PTPN1ALDH1A1PRSS12EDNRA
SCHEMBL4633874 0.85 ALDH1A1 (0.56) CXCR2MAPTALDH1A1MMP3RXFP1
SCHEMBL4635058 0.85 CXCR2 (0.58) CXCR2PTPN2PTPN1MAPTALDH1A1
SCHEMBL4633991 0.84 CXCR2 (0.62) CXCR2PTPN2PTPN1MAPTALDH1A1
SCHEMBL6652136 0.79 PTPN2 (0.52) CXCR2PTPN2PTPN1ALDH1A1MCL1
SCHEMBL4633952 0.79 CXCR2 (0.44) CXCR2MAPTALDH1A1MMP2MMP3
SCHEMBL4618003 0.78 CXCR2 (0.56) CXCR2MAPTALDH1A1LMNAPKM
SCHEMBL4633884 0.78 SENP2 (0.51) ALDH1A1EDNRA
SCHEMBL9024044 0.78 CXCR2 (0.54) CXCR2PTPN2PTPN1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685121-B1 ANTIDIABETIC COMPOUNDS COMPRISING BENZOTHIOPHENE DERIVATIVES MERCK PATENT GMBH (DE) 2008-06-11 EP claimed