SCHEMBL4634753

SCHEMBL4634753

CCc1nn(-c2ccncc2)c(Nc2ccc(Cl)cc2C(=O)O)c1-c1cccnc1F

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 8/20 0.43
ADORA2A P29274 1/20 0.39
ADORA2B P29275 1/20 0.39
DHODH Q02127 3/20 0.36
TGFBR1 P36897 2/20 0.36
FABP3 P05413 1/20 0.35
FABP4 P15090 1/20 0.35
MPO P05164 1/20 0.35
NR3C1 P04150 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM4E B2RXH2 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NUDT1 P36639 1/20 0.34
ACVR1B P36896 1/20 0.34
ACVRL1 P37023 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4666092 0.86 ADORA1 (0.46) ADORA1ADORA2AADORA2BFABP3FABP4
SCHEMBL4668225 0.84 ADORA1 (0.44) ADORA1ADORA2AADORA2BDHODHFABP3
SCHEMBL4633959 0.84 ADORA1 (0.44) ADORA1ADORA2AADORA2BDHODHTGFBR1
SCHEMBL4666257 0.80 ADORA1 (0.48) ADORA1DHODH
SCHEMBL14600439 0.80 ADORA1 (0.47) ADORA1DHODH
SCHEMBL14600188 0.79 ADORA1 (0.44) ADORA1ADORA2AADORA2BKDM4C
SCHEMBL14600260 0.76 DHODH (0.46) ADORA1DHODH
SCHEMBL4667046 0.74 ADORA1 (0.52) ADORA1ADORA2BFABP3FABP4KDM4C
SCHEMBL4668860 0.72 KCNMA1 (0.38) TGFBR1KDM4ENUDT1
SCHEMBL5090346 0.70 ADORA1 (0.59) ADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928455-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES Bayer Healthcare, LLC (US) 2008-06-11 EP disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed