SCHEMBL4637833

SCHEMBL4637833

CCOC(=O)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1cccnc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.59
SMN1; SMN2 Q16637 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
IDH1 O75874 1/20 0.43
CDC7 O00311 1/20 0.43
DBF4 Q9UBU7 1/20 0.43
MAPT P10636 1/20 0.41
PAX8 Q06710 1/20 0.40
GPBAR1 Q8TDU6 1/20 0.40
DCTPP1 Q9H773 1/20 0.39
KDR P35968 1/20 0.39
CACNA1B Q00975 1/20 0.39
APBA1 Q02410 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRA5 P31644 1/20 0.39
MMP2 P08253 1/20 0.39
MMP13 P45452 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637999 0.90 IDH1 (0.46) CYP19A1SMN1; SMN2KDM4EALDH1A1IDH1
SCHEMBL4637752 0.89 CYP19A1 (0.74) CYP19A1SMN1; SMN2ALDH1A1HPGDMAPT
SCHEMBL4639420 0.88 CYP19A1 (0.60) CYP19A1SMN1; SMN2KDM4EMAPTCACNA1B
SCHEMBL4637742 0.86 ALDH1A1 (0.52) CYP19A1ALDH1A1HPGDIDH1GPBAR1
SCHEMBL4637771 0.83 IDH1 (0.42) CYP19A1ALDH1A1IDH1MAPTGPBAR1
SCHEMBL4637730 0.83 MAPT (0.50) CYP19A1SMN1; SMN2KDM4EALDH1A1IDH1
SCHEMBL4637772 0.83 IDH1 (0.51) CYP19A1SMN1; SMN2KDM4EALDH1A1IDH1
SCHEMBL4638568 0.82 IDH1 (0.54) CYP19A1SMN1; SMN2KDM4EIDH1
SCHEMBL5797387 0.80 CYP19A1 (0.57) CYP19A1SMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL6071984 0.80 CYP19A1 (0.52) CYP19A1SMN1; SMN2KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed