SCHEMBL4638568

SCHEMBL4638568

COC(=O)c1nnn(Cc2ccc(C(F)(F)F)cc2)c1-c1cccnc1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.54
CYP19A1 P11511 5/20 0.49
SMN1; SMN2 Q16637 2/20 0.47
CYP1A2 P05177 1/20 0.47
HIF1A Q16665 5/20 0.43
EPAS1 Q99814 5/20 0.43
CFTR P13569 1/20 0.42
PTGER4 P35408 1/20 0.42
ADORA3 P0DMS8 1/20 0.41
DGAT2 Q96PD7 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637999 0.92 IDH1 (0.46) IDH1CYP19A1SMN1; SMN2CYP1A2CFTR
SCHEMBL4637730 0.90 MAPT (0.50) IDH1CYP19A1SMN1; SMN2CYP1A2PTGER4
SCHEMBL4638551 0.87 IDH1 (0.55) IDH1CYP19A1HIF1AEPAS1PTGER4
SCHEMBL4638983 0.86 IDH1 (0.49) IDH1CYP19A1HIF1AEPAS1PTGER4
SCHEMBL4637961 0.85 CFTR (0.46) IDH1CYP19A1SMN1; SMN2CFTRDGAT2
SCHEMBL4637734 0.85 CYP19A1 (0.46) IDH1CYP19A1SMN1; SMN2CYP1A2PTGER4
SCHEMBL4637971 0.84 CYP19A1 (0.50) IDH1CYP19A1SMN1; SMN2CYP1A2
SCHEMBL4637833 0.82 CYP19A1 (0.59) IDH1CYP19A1SMN1; SMN2KDM4E
SCHEMBL4637772 0.80 IDH1 (0.51) IDH1CYP19A1SMN1; SMN2CFTRKDM4E
SCHEMBL4707976 0.80 CYP19A1 (0.57) CYP19A1SMN1; SMN2CYP1A2ADORA3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed