SCHEMBL4637940

SCHEMBL4637940

CC(C)(C)[Si](C)(C)OCc1onc(-c2ccccc2Cl)c1C(=O)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.41
TACR1 P25103 1/20 0.37
ALDH1A1 P00352 2/20 0.36
GPBAR1 Q8TDU6 8/20 0.35
EPAS1 Q99814 2/20 0.35
MAPT P10636 2/20 0.34
MAPK1 P28482 1/20 0.34
RECQL P46063 1/20 0.34
TSHR P16473 2/20 0.34
HPGD P15428 1/20 0.34
ADORA3 P0DMS8 1/20 0.33
P2RX7 Q99572 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637783 0.93 TACR1 (0.41) TACR1ALDH1A1GPBAR1EPAS1MAPT
SCHEMBL4637701 0.93 GPBAR1 (0.38) IDH1TACR1ALDH1A1GPBAR1EPAS1
SCHEMBL4637809 0.90 EPAS1 (0.36) IDH1TACR1ALDH1A1GPBAR1EPAS1
SCHEMBL4637937 0.89 IDH1 (0.43) IDH1ALDH1A1GPBAR1EPAS1MAPT
SCHEMBL4637747 0.88 EPAS1 (0.38) TACR1ALDH1A1GPBAR1EPAS1MAPT
SCHEMBL4637782 0.87 IDH1 (0.42) IDH1ALDH1A1GPBAR1EPAS1MAPT
SCHEMBL4639007 0.86 GPBAR1 (0.37) IDH1TACR1ALDH1A1GPBAR1EPAS1
SCHEMBL4639367 0.84 TACR1 (0.32) TACR1GPBAR1EPAS1MAPT
SCHEMBL4638834 0.84 TACR1 (0.32) TACR1GPBAR1EPAS1MAPT
SCHEMBL4638539 0.83 IDH1 (0.40) IDH1ALDH1A1GPBAR1EPAS1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed