SCHEMBL4638834

SCHEMBL4638834

CC(C)(C)[Si](C)(C)OCc1onc(-c2cnccc2Cl)c1C(=O)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1Cl

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.32
GPBAR1 Q8TDU6 9/20 0.31
AKR1C3 P42330 1/20 0.30
TP53 P04637 1/20 0.30
MAPT P10636 1/20 0.30
EPAS1 Q99814 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4639367 0.94 TACR1 (0.32) TACR1GPBAR1AKR1C3TP53MAPT
SCHEMBL4637747 0.91 EPAS1 (0.38) TACR1GPBAR1TP53MAPTEPAS1
SCHEMBL4638040 0.89 ALDH1A1 (0.31) TACR1GPBAR1
SCHEMBL4639459 0.87 TACR1 (0.34) TACR1AKR1C3TP53MAPTEPAS1
SCHEMBL4637966 0.87 KMT2A (0.41) TACR1TP53MAPT
SCHEMBL4637701 0.85 GPBAR1 (0.38) TACR1GPBAR1MAPTEPAS1
SCHEMBL4637842 0.85 TACR1 (0.36) TACR1AKR1C3TP53MAPT
SCHEMBL4637940 0.84 IDH1 (0.41) TACR1GPBAR1MAPTEPAS1
SCHEMBL4637809 0.84 EPAS1 (0.36) TACR1GPBAR1MAPTEPAS1
SCHEMBL4637945 0.83 EPAS1 (0.37) TACR1GPBAR1TP53MAPTEPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed