SCHEMBL4637701

SCHEMBL4637701

CC(C)(C)[Si](C)(C)OCc1onc(-c2ccccc2Cl)c1C(=O)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccncc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 5/20 0.38
MAPT P10636 2/20 0.36
TACR1 P25103 1/20 0.36
RECQL P46063 1/20 0.36
EPAS1 Q99814 2/20 0.36
TSHR P16473 2/20 0.35
HPGD P15428 1/20 0.35
ALDH1A1 P00352 2/20 0.34
IDH1 O75874 1/20 0.34
CYP19A1 P11511 2/20 0.33
LMNA P02545 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
GRM2 Q14416 1/20 0.33
NLRP3 Q96P20 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637783 0.95 TACR1 (0.41) GPBAR1MAPTTACR1RECQLEPAS1
SCHEMBL4639007 0.93 GPBAR1 (0.37) GPBAR1MAPTTACR1RECQLEPAS1
SCHEMBL4637940 0.93 IDH1 (0.41) GPBAR1MAPTTACR1RECQLEPAS1
SCHEMBL4637809 0.90 EPAS1 (0.36) GPBAR1MAPTTACR1RECQLEPAS1
SCHEMBL4637747 0.90 EPAS1 (0.38) GPBAR1MAPTTACR1RECQLEPAS1
SCHEMBL6385074 0.87 GPBAR1 (0.39) GPBAR1MAPTTACR1RECQLEPAS1
SCHEMBL4638005 0.86 GPBAR1 (0.40) GPBAR1MAPTTACR1RECQLEPAS1
SCHEMBL4638834 0.85 TACR1 (0.32) GPBAR1MAPTTACR1EPAS1
SCHEMBL4639367 0.85 TACR1 (0.32) GPBAR1MAPTTACR1EPAS1
SCHEMBL4706457 0.83 ALDH1A1 (0.44) GPBAR1MAPTTACR1RECQLEPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed